Rankings / Muscle & Strength

Myostatin / activin-pathway inhibitors (non-bimagrumab)

Muscle & Strength · Myostatin/activin blockade

Tier C

wadamyostatinactivininvestigationalbanned-sport
4.9 / 10
Tier C
Ev 6.0 Bn 5.0 Sf 3.5

What this is

WADA coverage: activin A-neutralizing antibodies, activin receptor IIB competitors, decoy activin receptors, ACE-031, anti-activin receptor IIB antibodies, myostatin inhibitors, agents reducing or ablating myostatin expression, myostatin-binding proteins, follistatin, myostatin propeptide, myostatin- or precursor-neutralizing antibodies, apitegromab, domagrozumab, landogrozumab and stamulumab. Bimagrumab remains its own row. Additional WADA alias coverage: luspatercept and sotatercept are TGF-beta/activin-family ligand traps listed by WADA under related growth-factor modulation.

Mechanism

Blocking myostatin or activin receptor signaling can increase lean mass in some clinical contexts; functional improvements are much less consistent than muscle-volume changes.

Dose & route

Trial dosing varies widely by biologic; no approved enhancement dose

Citations

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This is an independent synthesis of published research by a non-clinician. Scores are opinions supported by citations, not prescriptions. See the full disclaimer and methodology for how this score was produced and what it does and doesn't mean.