Rankings / Cognitive

Solriamfetol (Sunosi)

Cognitive · DNRI / wakefulness-promoting

Tier B

dopaminednriadhdcontrolled-substanceprescriptionawaiting-readout
6.8 / 10
Tier B
Ev 8.0 Bn 8.0 Sf 5.0

What this is

Originally developed by Aerial BioPharma and Jazz Pharmaceuticals; **Axsome Therapeutics acquired Sunosi from Jazz in March 2022** and now drives the development program. Distinguishing pharmacology vs modafinil: direct dopamine + norepinephrine reuptake inhibition (closer to a mild amphetamine than to modafinil); preclinical mouse data show comparable wake-promotion but less anxiety-related behavior and lower locomotor activation than modafinil at equivalent wake-promoting doses. **Major 2025 development**: FOCUS Phase 3 in adult ADHD (Axsome press release March 25 2025) met primary endpoint at 150 mg (AISRS reduction -17.7 vs placebo -14.3; statistically significant; 53.5% response rate vs 41.3% placebo). Axsome announced sNDA preparation for the ADHD indication. SUSTAIN Phase 3 in shift work disorder ongoing with topline expected 2026. **Cardiovascular caveat**: dose-related SBP/DBP increases at peak (~2 hr post-dose) are transient across 24 hr at 150 mg/day, but the indicated populations all carry elevated baseline CV risk — small chronic BP elevations are clinically meaningful for MACE risk. 2024 FAERS retrospective pharmacovigilance (Q3 2019 – Q1 2024) identified 30 disproportionality signals; AE profile consistent with label. Real-world preference: in a 62-patient retrospective, 71% of patients preferred solriamfetol over modafinil/armodafinil after switching; 29% reverted. Distinct from Pitolisant (Wakix) — the only non-scheduled wakefulness Rx — see adjacent row.

Mechanism

Selective dopamine and norepinephrine reuptake inhibitor (DNRI); mechanistically distinct from modafinil's adenosine/orexin pathway; FDA-approved 2019 for excessive daytime sleepiness in narcolepsy and OSA; March 2025 FOCUS Phase 3 also positive in adult ADHD

Dose & route

75-150 mg PO once daily (FOCUS Ph3 300 mg dose was numerically superior but NOT statistically significant on primary)

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